An androgenic agent, contains testosterone esters. It affects the development and function of the external
genitalia, prostate, seminal vesicles, and secondary sexual
characteristics (voice, hair). Participates in the formation of the constitution of the body and sexual
behavior, activates libido and potency, stimulates spermatogenesis. It is an antagonist of the female sex hormones-estrogens. It has an anabolic effect, which is manifested in the stimulation of protein synthesis, the delay necessary for the synthesis of protein, potassium, sulfur, phosphorus, which enhance the fixation of calcium in the bones and increase the muscle mass of the body. Testosterone esters have different rates of absorption and excretion, which
ensures a rapid development of the effect and a long-lasting effect (up to 4 weeks) after a single administration.
An androgenic agent, it also has an anabolic effect. In target cells (skin, prostate, seminal vesicles, epididymus), 5-alpha-reductase is reduced to 5-alpha-dihydrotestosterone, which specifically interacts with membrane receptors on the cell surface and penetrates into the nucleus. In some tissues (including the hypothalamus) turns into estradiol.
In men, it stimulates the development and activity of the gonads, prostate gland, seminal vesicles, the formation of secondary male characteristics (growth, low voice, beard and mustache growth), increases libido and potency; indirectly, through the central nervous system, it affects sexual behavior.
Reduces the deposition of fat and the excretion of trace elements. Inhibits the production and release of LH and FSH by the pituitary gland.
It has anabolic effects: participates in the growth of the skeleton, increases the mass of skeletal muscles; causes the retention of nitrogen, phosphorus, K+ and sulfur, which are necessary for protein synthesis.
The testosterone esters that are part of the drug have different rates of absorption and excretion, which ensures a rapid development of the effect and a long-lasting effect (up to 4 weeks) after a single injection: testosterone propionate acts during the first day, phenylpropionate and isocapronate-24 hours after the injection.
Dosage and course of treatment
In / m. Men-100-200 mg 1 time in 15 days, the course of treatment-10-15 injections; for impotence and menopausal syndrome-0.1 g 1 time in 15 days, the course of treatment - 5 injections.
Women with menopausal syndrome are prescribed 0.1 g 1 time in 2-3 weeks; for breast and ovarian cancer-100-200 mg after 1-2 weeks, treatment is long-term.
|Active ingredient, mg||250|
|1 bottle, ml||10|
|Bottles in the package, pcs||1|